187 results on '"Saulnier, Mark"'
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2. The discovery of BMS-737 as a potent, CYP17 lyase-selective inhibitor for the treatment of castration-resistant prostate cancer
3. Discovery and Preclinical Profiling of GSK3839919, a Potent HIV-1 Allosteric Integrase Inhibitor
4. SNAr reactions of 5-bromo-2-chloro-4-fluoro-3-iodopyridine and its 3-substituted analogs
5. Biochemical and transcriptional profiling to triage additional activities in a series of IGF-1R/IR inhibitors
6. 5-Bromo-2-chloro-4-fluoro-3-iodopyridine as a Halogen-rich Intermediate for the Synthesis of Pentasubstituted Pyridines
7. Anti-Tumor Effects of Antibody--Alkaline Phosphatase Conjugates in Combination with Etoposide Phosphate
8. Synthesis of new pyrrolo[3,4-b]indol-3-ones as latent substrates for pyrrolo[3,4-b]indoles
9. 5-Bromo-2-chloro-4-fluoro-3-iodopyridine as a Halogen-rich Intermediate for the Synthesis of Pentasubstituted Pyridines.
10. Chapter 5.5 Five-membered ring systems: With N and S (Se) atoms
11. The Synthesis of Structurally Novel Bridged Glycosidic Fluoroindolocarbazoles as Topoisomerase I Inhibitors
12. Quantitation of the interaction of the immunosuppressant deoxyspergualin and analogs with Hsc70 and Hsp90
13. Preclinical antitumor activity of a soluble etoposide analog, BMY-40481-30
14. A Practical Approach for Enantio- and Diastereocontrol in the Synthesis of 2,3-Disubstituted Succinic Acid Esters: Synthesis of the pan-Notch Inhibitor BMS-906024
15. Syntheses and Diels-Alder cycloaddition reactions of 4H-furo(3,4-b)indoles: a regiospecific Diels-Alder synthesis of ellipticine
16. A versatile and efficient construction of the 6H-pyrido(4,3-b)carbazole ring system: synthesis of the antitumor alkaloids ellipticine, 9-methoxyellipticine, and olivacine and their analogues
17. Synthesis of new pyrrolo[3,4-b]indol-3-ones as latent substrates for pyrrolo[3,4-b]indoles.
18. Insulin-like growth factor-1 receptor (IGF-1R) kinase inhibitors: SAR of a series of 3-[6-(4-substituted-piperazin-1-yl)-4-methyl-1H-benzimidazol-2-yl]-1H-pyridine-2-one
19. Nucleophilic Capture of the Imino-Quinone Methide Type Intermediates Generated from 2-Aminothiazol-5-yl Carbinols
20. Balancing oral exposure with Cyp3A4 inhibition in benzimidazole-based IGF-IR inhibitors
21. Novel Indole Chemistry in the Synthesis of Heterocycles
22. Tumor Development by Transgenic Expression of a Constitutively Active Insulin-Like Growth Factor I Receptor
23. Discovery of a Fluoroindolo[2,3-a]carbazole Clinical Candidate with Broad Spectrum Antitumor Activity in Preclinical Tumor Models Superior to the Marketed Oncology Drug, CPT-11
24. Design and Synthesis of a Fluoroindolocarbazole Series as Selective Topoisomerase I Active Agents. Discovery of Water-Soluble 3,9-Difluoro-12,13-dihydro-13-[6-amino-β- <scp>d</scp>-glucopyranosyl]-5H,13H-benzo[b]- thienyl[2,3-a]pyrrolo[3,4-c]carbazole- 5,7(6H)-dione (BMS-251873) with Curative Antitumor Activity against Prostate Carcinoma Xenograft Tumor Model
25. Intramolecular Diels-Alder Reactions of 4H-Furo[3,4-b]indoles. New Syntheses of Benzo[a]carbazoles and Benzo[c]carbazoles
26. A Practical Approach for Enantio- and Diastereocontrol in the Synthesis of 2,3-Disubstituted Succinic Acid Esters: Synthesis of the pan-Notch Inhibitor BMS-906024
27. Microwave-assisted synthesis of primary amine HX salts from halides and 7 M ammonia in methanol
28. Synthesis of etoposide phosphate, BMY-40481: A water-soluble clinically active prodrug of etoposide
29. An efficient method for the synthesis of guanidino prodrugs
30. Quantitation of the Interaction of the Immunosuppressant Deoxyspergualin and Analogs with Hsc70 and Hsp90
31. Biochemical and transcriptional profiling to triage additional activities in a series of IGF-1R/IR inhibitors
32. Synthesis and biological activity of 3′,4′,5′-trihydroxy etoposide
33. Synthesis of tritium labeled (±) 15-deoxyspergualin trihydrochloride
34. ChemInform Abstract: An Unusual Oxidative Cyclization. A Synthesis and Absolute Stereochemical Assignment of (-)-Rocaglamide
35. ChemInform Abstract: A Versatile and Efficient Construction of the 6H-Pyrido(4,3-b) carbazole Ring System. Syntheses of the Antitumor Alkaloids Ellipticine, 9-Methoxyellipticine, and Olivacine and Their Analogues
36. ChemInform Abstract: Syntheses of 2,3-Dihalo-1-(phenylsulfonyl)indoles (IV), (VI)
37. ChemInform Abstract: Regioselective ortho-Lithiation of Halopyridines. Synthesis of ortho- Disubstituted Pyridines and a Convenient Generation of 3,4-Pyridyne
38. ChemInform Abstract: Syntheses and Diels-Alder Cycloaddition Reactions of 4H-Furo(3,4-b) indoles. A Regiospecific Diels-Alder Synthesis of Ellipticine
39. ChemInform Abstract: An Efficient Method for the Synthesis of Guanidino Prodrugs
40. ChemInform Abstract: Synthesis of a Rebeccamycin-Related Indolo(2,3-a)carbazole by Palladium(0)-Catalyzed Polyannulation
41. ChemInform Abstract: Intramolecular Diels-Alder Reactions of 4H-Furo[3,4-b]indoles. New Syntheses of Benzo[a]carbazoles and Benzo[c]carbazoles
42. ChemInform Abstract: Nucleophilic Capture of the Imino-Quinone Methide Type Intermediates Generated from 2-Aminothiazol-5-yl Carbinols
43. SYNTHESES OF 2,3-DIHALO-1-(PHENYLSULFONYL)INDOLES
44. Synthesis of biological evaluation of 4′-deshydroxy-4′-methyl etoposide and teniposide analogs
45. Syntheses and Diels-Alder cycloaddition reactions of 4H-furo[3,4-b]indoles. A regiospecific Diels-Alder synthesis of ellipticine
46. Etoposide(VP16): Chemical reactivity of etoposide ortho-quinone with amines and thiols
47. SAR of PXR transactivation in benzimidazole-based IGF-1R kinase inhibitors
48. Discovery of a 2,4-disubstituted pyrrolo[1,2-f][1,2,4]triazine inhibitor (BMS-754807) of insulin-like growth factor receptor (IGF-1R) kinase in clinical development
49. Preclinical antitumor activity of a soluble etoposide analog, BMY-40481-30
50. 2-(1H-Imidazol-4-yl)ethanamine and 2-(1H-pyrazol-1-yl)ethanamine side chain variants of the IGF-1R inhibitor BMS-536924
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