124 results on '"Raheem, Izzat"'
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2. To Market, to Market—2020: Small Molecules
3. Structural understanding of non-nucleoside inhibition in an elongating herpesvirus polymerase
4. Cerastecin Inhibition of the Lipooligosaccharide Transporter MsbA to Combat Acinetobacter baumannii: From Screening Impurity to In VivoEfficacy
5. Stabilized trimeric peptide immunogens of the complete HIV-1 gp41 N-heptad repeat and their use as HIV-1 vaccine candidates.
6. To Market, to Market—2019: Small Molecules
7. Discovery of MK-8189, a Highly Potent and Selective PDE10A Inhibitor for the Treatment of Schizophrenia
8. Preclinical Characterization of the Phosphodiesterase 10A PET Tracer [11C]MK-8193
9. The novel phosphodiesterase 10A inhibitor THPP-1 has antipsychotic-like effects in rat and improves cognition in rat and rhesus monkey
10. P546. Preclinical Characterization and Phase 1 Evaluation of the Tolerability, Pharmacokinetics, and Enzyme Occupancy of MK-8189, a Novel PDE10A Inhibitor
11. Building a Culture of Medicinal Chemistry Knowledge Sharing
12. Genetic deletion and pharmacological inhibition of phosphodiesterase 10A protects mice from diet-induced obesity and insulin resistance
13. Stark spectroscopy of size-selected helical H-aggregates of a cyanine dye templated by duplex DNA. Effect of exciton coupling on electronic polarizabilities
14. Characterization of chiral H and J aggregates of cyanine dyes formed by DNA templating using stark and fluorescence spectroscopies
15. Discovery and optimization of 2-pyridinone aminal integrase strand transfer inhibitors for the treatment of HIV
16. Discovery of pyrazolopyrimidine phosphodiesterase 10A inhibitors for the treatment of schizophrenia
17. Synthesis and Antiviral Evaluation of Carbocyclic Nucleoside Analogs of Nucleoside Reverse Transcriptase Translocation Inhibitor MK-8591 (4′-Ethynyl-2-fluoro-2′-deoxyadenosine)
18. Discovery of [11C]MK-8193 as a PET tracer to measure target engagement of phosphodiesterase 10A (PDE10A) inhibitors
19. Catalytic asymmetric total syntheses of quinine and quinidine
20. Discovery of tetrahydropyridopyrimidine phosphodiesterase 10A inhibitors for the treatment of schizophrenia
21. Enantioselective Pictet-Spengler-type cyclizations of hydroxylactams: H-bond donor catalysis by anion binding
22. Correction to Discovery of 2-Pyridinone Aminals: A Prodrug Strategy to Advance a Second Generation of HIV-1 Integrase Strand Transfer Inhibitors
23. Preclinical Characterization of the Phosphodiesterase 10A PET Tracer [11C]MK-8193
24. Discovery of [ 11 C ] MK - 8193 as a PET tracer to measure target engagement of phosphodiesterase 10A (PDE10A) inhibitors
25. Discovery of 2-Pyridinone Aminals: A Prodrug Strategy to Advance a Second Generation of HIV-1 Integrase Strand Transfer Inhibitors
26. Discovery of piperidine ethers as selective orexin receptor antagonists (SORAs) inspired by filorexant
27. Efficient synthesis of highly functionalized tetrahydropyridopyrimidines by a novel three-component coupling reaction
28. ChemInform Abstract: Sustainable Chromatography (an Oxymoron?)
29. Sustainable chromatography (an oxymoron?)
30. Genetic Deletion and Pharmacological Inhibition of Phosphodiesterase 10A Protects Mice From Diet-Induced Obesity and Insulin Resistance
31. Merck’s Reaction Review Policy: An Exercise in Process Safety
32. ChemInform Abstract: Sustainable Practices in Medicinal Chemistry: Current State and Future Directions
33. Sustainable Practices in Medicinal Chemistry: Current State and Future Directions
34. ChemInform Abstract: C—O Cross‐Coupling of Activated Aryl and Heteroaryl Halides with Aliphatic Alcohols.
35. ChemInform Abstract: Discovery of Tetrahydropyridopyrimidine Phosphodiesterase 10A Inhibitors for the Treatment of Schizophrenia.
36. CO Cross-Coupling of Activated Aryl and Heteroaryl Halides with Aliphatic Alcohols
37. ChemInform Abstract: Efficient Synthesis of Highly Functionalized Tetrahydropyridopyrimidines by a Novel Three‐Component Coupling Reaction.
38. ChemInform Abstract: Regio- and Enantioselective Catalytic Cyclization of Pyrroles onto N-Acyliminium Ions.
39. Regio- and Enantioselective Catalytic Cyclization of Pyrroles onto N-Acyliminium Ions
40. ChemInform Abstract: Enantioselective Pictet—Spengler‐Type Cyclizations of Hydroxylactams: H‐Bond Donor Catalysis by Anion Binding.
41. Enantioselective Pictet−Spengler-Type Cyclizations of Hydroxylactams: H-Bond Donor Catalysis by Anion Binding
42. Highly Enantioselective Aza-Baylis-Hillman Reactions Catalyzed by Chiral Thiourea Derivatives
43. Catalytic Asymmetric Total Syntheses of Quinine and Quinidine
44. Merck’sReaction Review Policy: An Exercise in Process Safety.
45. SustainablePractices in Medicinal Chemistry: CurrentState and Future Directions.
46. Antiviral Prodrugs Of Tenofovir
47. Preclinical Evaluation of MK-8189: A Novel Phosphodiesterase 10A Inhibitor for the Treatment of Schizophrenia.
48. Discovery of Broad-Spectrum Herpes Antiviral Oxazolidinone Amide Derivatives and Their Structure-Activity Relationships.
49. Stabilized trimeric peptide immunogens of the complete HIV-1 gp41 N-heptad repeat and their use as HIV-1 vaccine candidates.
50. Correction to Discovery of 2-Pyridinone Aminals: A Prodrug Strategy to Advance a Second Generation of HIV-1 Integrase Strand Transfer Inhibitors.
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