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One-Pot, Three-Component Assembly of Indoloquinolines: Total Synthesis of Isocryptolepine

Authors :
Aksenov, Alexander A.V.
Rubin, Michael
Aksenov, Dmitrii D.A.
Orazova, Naila N.A.
Aksenov, Nicolai N.A.
Griaznov, Georgii G.D.
De Carvalho, Annelise
Kiss, Robert
Mathieu, Véronique
Kornienko, Alexander
Aksenov, Alexander A.V.
Rubin, Michael
Aksenov, Dmitrii D.A.
Orazova, Naila N.A.
Aksenov, Nicolai N.A.
Griaznov, Georgii G.D.
De Carvalho, Annelise
Kiss, Robert
Mathieu, Véronique
Kornienko, Alexander
Source :
Journal of organic chemistry, 82 (6
Publication Year :
2017

Abstract

Indolo[3,2-c]quinolones have been efficiently synthesized via an acid-mediated, one-pot, three-component condensation of arylhydrazines, o-aminoacetophenones, and triazines or nitriles. The synthetic application of this method is showcased by the concise synthesis of isocryptolepine alkaloid and a series of its synthetic analogues with demonstrated cancer cell antiproliferative activities.<br />SCOPUS: ar.j<br />info:eu-repo/semantics/published

Details

Database :
OAIster
Journal :
Journal of organic chemistry, 82 (6
Notes :
No full-text files, English
Publication Type :
Electronic Resource
Accession number :
edsoai.ocn994546631
Document Type :
Electronic Resource