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Mucolytic Agents Can Enhance HER2 Receptor Accessibility for [(89)Zr]Trastuzumab, Improving HER2 Imaging in a Mucin-Overexpressing Breast Cancer Xenograft Mouse Model.

Authors :
Wimana, Zéna
Gebhart, Géraldine
Guiot, Thomas
Vanderlinden, Bruno
Morandini, Renato
Doumont, Gilles
Sherer, Félicie
Van Simaeys, Gaëtan
Goldman, Serge
Ghanem, Ghanem Elias
Flamen, Patrick
Wimana, Zéna
Gebhart, Géraldine
Guiot, Thomas
Vanderlinden, Bruno
Morandini, Renato
Doumont, Gilles
Sherer, Félicie
Van Simaeys, Gaëtan
Goldman, Serge
Ghanem, Ghanem Elias
Flamen, Patrick
Source :
Molecular imaging and biology
Publication Year :
2015

Abstract

Binding of trastuzumab to HER2 receptors can be impaired by steric hindrance caused by mucin MUC4. As mucolytic drugs can breakdown disulfide bonds of mucoproteins, we checked if this approach could positively affect zirconium-89-labeled trastuzumab ([(89)Zr]T) binding/uptake.<br />SCOPUS: ar.j<br />info:eu-repo/semantics/published

Details

Database :
OAIster
Journal :
Molecular imaging and biology
Notes :
1 full-text file(s): application/pdf, English
Publication Type :
Electronic Resource
Accession number :
edsoai.ocn915541237
Document Type :
Electronic Resource