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POTENTIAL ANTIMALARIALS STRUCTURALLY RELATED TO QUININE.

Authors :
COLORADO UNIV BOULDER
Coffen,David L.
COLORADO UNIV BOULDER
Coffen,David L.
Source :
DTIC AND NTIS
Publication Year :
1969

Abstract

The base-catalyzed condensation of 3-quinuclidinone with quinoline carboxaldehydes provides easy access to a large number of compounds which may be loosely described as desvinylquinine derivatives. Many such substances have been synthesized and submitted for antimalarial screening. Of particular interest are the quinolinemethanols obtained by acid-catalyzed hydration of the condensation products. The unique metal complexes of 2-(2'-quinolyl)methylene-3-quinuclidinone which were encountered during this work and progress on an attempt to synthesize the complete quinine skeleton are also described. (Author)

Details

Database :
OAIster
Journal :
DTIC AND NTIS
Notes :
text/html, English
Publication Type :
Electronic Resource
Accession number :
edsoai.ocn831485884
Document Type :
Electronic Resource