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The small molecule CLP257 does not modify activity of the K+-Cl- co-transporter KCC2 but does potentiate GABAA receptor activity

Authors :
Cardarelli, Ross A
Jones, Karen
Pisella, Lucie I
Wobst, Heike J
McWilliams, Lisa J
Sharpe, Paul M
Burnham, Matthew P
Baker, David J
Chudotvorova, Ilona
Guyot, Justine
Silayeva, Liliya
Morrow, Danielle H
Dekker, Niek
Zicha, Stephen
Davies, Paul A
Holenz, Jörg
Duggan, Mark E
Dunlop, John
Mather, Robert J
Wang, Qi
Medina, Igor
Brandon, Nicholas J
Deeb, Tarek Z
Moss, Stephen J
Source :
Nature Medicine. December 2017, Vol. 23 Issue 12, p1394, 3 p.
Publication Year :
2017

Abstract

Author(s): Ross A Cardarelli [1, 10]; Karen Jones [2, 10]; Lucie I Pisella [3, 4, 10]; Heike J Wobst [1, 5]; Lisa J McWilliams [6]; Paul M Sharpe [2]; Matthew [...]

Details

Language :
English
ISSN :
10788956
Volume :
23
Issue :
12
Database :
Gale General OneFile
Journal :
Nature Medicine
Publication Type :
Academic Journal
Accession number :
edsgcl.517771180
Full Text :
https://doi.org/10.1038/nm.4442