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Tandem application of virtual screening and NMR experiments in the discovery of brand new DNA quadruplex groove binders

Authors :
Cosconati, Sandro
Marinelli, Luciana
Trotta, Roberta
Virno, Ada
Mayol, Luciano
Novellino, Ettore
Olson, Arthur J.
Randazzo, Antonio
Source :
Journal of the American Chemical Society. Nov 18, 2009, Vol. 131 Issue 45, 16336-16337
Publication Year :
2009

Abstract

A structure-based virtual screening campaign is performed by using the X-ray structure of the [[d(TGGGGT)].sub.4] quadruplex with the aim of detecting new and structurally diverse groove binders. Six brand new different molecular entities have interacted with the groove through NMR experiments.

Details

Language :
English
ISSN :
00027863
Volume :
131
Issue :
45
Database :
Gale General OneFile
Journal :
Journal of the American Chemical Society
Publication Type :
Academic Journal
Accession number :
edsgcl.213334162