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Discovery of small molecule agonists of the Relaxin Family Peptide Receptor 2

Authors :
Maria Esteban-Lopez
Kenneth J. Wilson
Courtney Myhr
Elena M. Kaftanovskaya
Mark J. Henderson
Noel T. Southall
Xin Xu
Amy Wang
Xin Hu
Elena Barnaeva
Wenjuan Ye
Emmett R. George
John T. Sherrill
Marc Ferrer
Roy Morello
Irina U. Agoulnik
Juan J. Marugan
Alexander I. Agoulnik
Source :
Communications Biology, Vol 5, Iss 1, Pp 1-12 (2022)
Publication Year :
2022
Publisher :
Nature Portfolio, 2022.

Abstract

Specific small molecule RXFP2 agonists with favorable pharmacokinetic properties induce gubernacular invagination in mouse embryos, increase mineralization activity in human osteoblasts in vitro, and improve bone trabecular parameters in adult mice.

Subjects

Subjects :
Biology (General)
QH301-705.5

Details

Language :
English
ISSN :
23993642
Volume :
5
Issue :
1
Database :
Directory of Open Access Journals
Journal :
Communications Biology
Publication Type :
Academic Journal
Accession number :
edsdoj.50c86baebeb04e3ebabf87beea0be0a0
Document Type :
article
Full Text :
https://doi.org/10.1038/s42003-022-04143-9