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Quinoline-3-carboxamide Derivatives as Potential Cholesteryl Ester Transfer Protein Inhibitors

Authors :
Jing-Kang Shen
Mao-Sheng Cheng
Yu-Fang Shi
Zhi-Heng Yang
Chao Yu
Pei-Wei Fan
Wen-Yan Li
Xu-Qiong Xiong
Dong-Mei Zhao
Source :
Molecules, Vol 17, Iss 5, Pp 5497-5507 (2012)
Publication Year :
2012
Publisher :
MDPI AG, 2012.

Abstract

A series of novel quinoline-3-carboxamide derivatives 10–17 and 23–27 were designed and synthesized as cholesteryl ester transfer protein (CETP) inhibitors. All of them exhibited activity against CETP. Particularly, compounds 24 and 26 displayed the best activity against CETP with the same inhibitory rate of 80.1%.

Details

Language :
English
ISSN :
14203049 and 04538870
Volume :
17
Issue :
5
Database :
Directory of Open Access Journals
Journal :
Molecules
Publication Type :
Academic Journal
Accession number :
edsdoj.2e2c756af0d045388703262bfa020eb1
Document Type :
article
Full Text :
https://doi.org/10.3390/molecules17055497