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The new-generation selective ROS1/NTRK inhibitor DS-6051b overcomes crizotinib resistant ROS1-G2032R mutation in preclinical models

Authors :
Ryohei Katayama
Bo Gong
Noriko Togashi
Masaya Miyamoto
Masaki Kiga
Shiho Iwasaki
Yasuki Kamai
Yuichi Tominaga
Yasuyuki Takeda
Yoshiko Kagoshima
Yuki Shimizu
Yosuke Seto
Tomoko Oh-hara
Sumie Koike
Naoki Nakao
Hiroyuki Hanzawa
Kengo Watanabe
Satoshi Yoda
Noriko Yanagitani
Aaron N. Hata
Alice T. Shaw
Makoto Nishio
Naoya Fujita
Takeshi Isoyama
Source :
Nature Communications, Vol 10, Iss 1, Pp 1-12 (2019)
Publication Year :
2019
Publisher :
Nature Portfolio, 2019.

Abstract

The treatment of ROS1-rearranged non-small cell lung cancer with the TKI crizotinib is limited due to the emergence of resistance. Here, the authors develop a new ROS1/NTRK inhibitor, DS-6051b, which overcomes crizotinib resistance in preclinical models.

Subjects

Subjects :
Science

Details

Language :
English
ISSN :
20411723
Volume :
10
Issue :
1
Database :
Directory of Open Access Journals
Journal :
Nature Communications
Publication Type :
Academic Journal
Accession number :
edsdoj.1fb146a2c258459e81f631757ffb5a98
Document Type :
article
Full Text :
https://doi.org/10.1038/s41467-019-11496-z