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Unraveling topoisomerase IA gate dynamics in presence of PPEF and its preclinical evaluation against multidrug-resistant pathogens

Authors :
Vikas Maurya
Raja Singh
Reman Kumar Singh
Stuti Pandey
Pooja Yadav
Palak Parashar
Rajni Gaind
Kshatresh Dutta Dubey
G. Naresh Patwari
Vibha Tandon
Source :
Communications Biology, Vol 6, Iss 1, Pp 1-20 (2023)
Publication Year :
2023
Publisher :
Nature Portfolio, 2023.

Abstract

Two potent inhibitors PPEF and BPVF of bacterial TopoIA enzymes function by impairing DNA binding and thus DNA cleavage and relaxation activities of bacterial topoisomerase I enzymes.

Subjects

Subjects :
Biology (General)
QH301-705.5

Details

Language :
English
ISSN :
23993642
Volume :
6
Issue :
1
Database :
Directory of Open Access Journals
Journal :
Communications Biology
Publication Type :
Academic Journal
Accession number :
edsdoj.1d3a56edcbf6496f947aa4da52ad7627
Document Type :
article
Full Text :
https://doi.org/10.1038/s42003-023-04412-1