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Discovery of 'Molecular Switches' within a Series of mGlu5 Allosteric Ligands Driven by a 'Magic Methyl' Effect Affording Both PAMs and NAMs with In Vivo Activity, Derived from an M1 PAM Chemotype
- Source :
- ACS Bio & Med Chem Au, Vol 1, Iss 1, Pp 21-30 (2021)
- Publication Year :
- 2021
- Publisher :
- American Chemical Society, 2021.
- Subjects :
- Biology (General)
QH301-705.5
Biochemistry
QD415-436
Subjects
Details
- Language :
- English
- ISSN :
- 26942437
- Volume :
- 1
- Issue :
- 1
- Database :
- Directory of Open Access Journals
- Journal :
- ACS Bio & Med Chem Au
- Publication Type :
- Academic Journal
- Accession number :
- edsdoj.1962d9086d84ecabe40eff8d58cb02f
- Document Type :
- article
- Full Text :
- https://doi.org/10.1021/acsbiomedchemau.1c00024