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Discovery of 'Molecular Switches' within a Series of mGlu5 Allosteric Ligands Driven by a 'Magic Methyl' Effect Affording Both PAMs and NAMs with In Vivo Activity, Derived from an M1 PAM Chemotype

Authors :
Lisa Barbaro
Alice L. Rodriguez
Ashlyn N. Blevins
Jonathan W. Dickerson
Natasha Billard
Olivier Boutaud
Jerri L. Rook
Colleen M. Niswender
P.Jeffrey Conn
Darren W. Engers
Craig W. Lindsley
Source :
ACS Bio & Med Chem Au, Vol 1, Iss 1, Pp 21-30 (2021)
Publication Year :
2021
Publisher :
American Chemical Society, 2021.

Details

Language :
English
ISSN :
26942437
Volume :
1
Issue :
1
Database :
Directory of Open Access Journals
Journal :
ACS Bio & Med Chem Au
Publication Type :
Academic Journal
Accession number :
edsdoj.1962d9086d84ecabe40eff8d58cb02f
Document Type :
article
Full Text :
https://doi.org/10.1021/acsbiomedchemau.1c00024