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TAS1553, a small molecule subunit interaction inhibitor of ribonucleotide reductase, exhibits antitumor activity by causing DNA replication stress

Authors :
Hiroyuki Ueno
Takuya Hoshino
Wakako Yano
Sayaka Tsukioka
Takamasa Suzuki
Shoki Hara
Yoshio Ogino
Khoon Tee Chong
Tatsuya Suzuki
Shingo Tsuji
Hikaru Itadani
Ikuo Yamamiya
Yoshihiro Otsu
Satoshi Ito
Toshiya Yonekura
Miki Terasaka
Nozomu Tanaka
Seiji Miyahara
Source :
Communications Biology, Vol 5, Iss 1, Pp 1-12 (2022)
Publication Year :
2022
Publisher :
Nature Portfolio, 2022.

Abstract

A small-molecule protein-protein interaction inhibitor of ribonucleotide reductase subunit, TAS1553, is shown to inhibit growth of both hematological and solid cancer xenograft tumors following oral administration in mice.

Subjects

Subjects :
Biology (General)
QH301-705.5

Details

Language :
English
ISSN :
23993642
Volume :
5
Issue :
1
Database :
Directory of Open Access Journals
Journal :
Communications Biology
Publication Type :
Academic Journal
Accession number :
edsdoj.06c93c29221d4c129be884628c9ba09b
Document Type :
article
Full Text :
https://doi.org/10.1038/s42003-022-03516-4