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Design and Characterization of a Natural Arf-GEFs Inhibitor Prodrug
- Source :
- Journal of medicinal chemistry. 65(18)
- Publication Year :
- 2022
-
Abstract
- Brefeldin A (BFA), a well-known natural Arf-GEFs inhibitor, is effective against hepatocellular carcinoma (HCC), while the poor solubility, serious toxicity, and short half-life limit its potential. Herein, distinct corresponding prodrugs of BFA, including esters
Details
- ISSN :
- 15204804
- Volume :
- 65
- Issue :
- 18
- Database :
- OpenAIRE
- Journal :
- Journal of medicinal chemistry
- Accession number :
- edsair.pmid..........a6f106343e693b88a38ebdd87ea6ddcd