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Identification of Thieno[3,2
- Source :
- Journal of medicinal chemistry. 64(16)
- Publication Year :
- 2021
-
Abstract
- Focal adhesion kinase (FAK) is overexpressed in highly invasive and metastatic cancers. To identify novel FAK inhibitors, we designed and synthesized various thieno[3,2
- Subjects :
- Mice, Inbred BALB C
Molecular Structure
Mice, Nude
Antineoplastic Agents
Thiophenes
Xenograft Model Antitumor Assays
Molecular Docking Simulation
Structure-Activity Relationship
Pyrimidines
fms-Like Tyrosine Kinase 3
Cell Line, Tumor
Focal Adhesion Kinase 1
Neoplasms
Animals
Humans
Female
Drug Screening Assays, Antitumor
Neoplasm Metastasis
Phosphorylation
Protein Kinase Inhibitors
Subjects
Details
- ISSN :
- 15204804
- Volume :
- 64
- Issue :
- 16
- Database :
- OpenAIRE
- Journal :
- Journal of medicinal chemistry
- Accession number :
- edsair.pmid..........7d6d1b1ab771cdc85d913f2784350fce