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Absorption, distribution, metabolism and excretion of darolutamide (a novel non-steroidal androgen receptor antagonist) in rats
- Source :
- Xenobiotica; the fate of foreign compounds in biological systems. 50(8)
- Publication Year :
- 2020
-
Abstract
- 1. Darolutamide is a novel selective androgen receptor antagonist consisting of two pharmacologically equipotent diastereoisomers. The absorption, distribution, metabolism and excretion properties of darolutamide in rats are reported.2. Non- or [
- Subjects :
- Health, Toxicology and Mutagenesis
Administration, Oral
Biological Availability
Absorption (skin)
Pharmacology
Toxicology
Blood–brain barrier
030226 pharmacology & pharmacy
Biochemistry
Excretion
03 medical and health sciences
Feces
0302 clinical medicine
Pharmacokinetics
medicine
Androgen Receptor Antagonists
Distribution (pharmacology)
Animals
Bile
Tissue Distribution
Chemistry
Diastereomer
General Medicine
Metabolism
Body Fluids
Rats
medicine.anatomical_structure
Darolutamide
Intestinal Absorption
030220 oncology & carcinogenesis
Pyrazoles
Subjects
Details
- ISSN :
- 13665928
- Volume :
- 50
- Issue :
- 8
- Database :
- OpenAIRE
- Journal :
- Xenobiotica; the fate of foreign compounds in biological systems
- Accession number :
- edsair.doi.dedup.....fc07f906daf87c912ef246192fe07225