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Exploiting furan's versatile reactivity in reversible and irreversible orthogonal peptide labeling

Authors :
Annemieke Madder
Dieter Buyst
Kurt Hoogewijs
Johan M. Winne
José C. Martins
Source :
Chemical communications (Cambridge, England). 49(28)
Publication Year :
2013

Abstract

A general method for the facile and versatile decoration of peptides is proposed exploiting furan based cycloaddition and electrophilic aromatic substitution reactions. Given the commercial availability of furylalanine derivatives for peptide synthesis, the current work significantly enlarges the toolbox of available methodologies for site specific labeling and conjugation of peptide probes.

Details

ISSN :
1364548X
Volume :
49
Issue :
28
Database :
OpenAIRE
Journal :
Chemical communications (Cambridge, England)
Accession number :
edsair.doi.dedup.....bd1c138e3c3bc8e968c8fd5a23d8a94a