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Atropisomeric Derivatives of 2‘,6‘-Disubstituted (R)-11-Phenylaporphine: Selective Serotonin 5-HT7 Receptor Antagonists
- Source :
- Journal of Medicinal Chemistry. 44:1337-1340
- Publication Year :
- 2001
- Publisher :
- American Chemical Society (ACS), 2001.
- Subjects :
- Aporphines
Stereochemistry
Molecular Conformation
CHO Cells
In Vitro Techniques
Crystallography, X-Ray
Binding, Competitive
Chemical synthesis
Structure-Activity Relationship
Cricetinae
Drug Discovery
Cyclic AMP
Animals
Receptor
5-HT receptor
Chemistry
Antagonist
Brain
Stereoisomerism
In vitro
Rats
Receptors, Serotonin
Benzene derivatives
Molecular Medicine
Serotonin Antagonists
Serotonin
Selectivity
Subjects
Details
- ISSN :
- 15204804 and 00222623
- Volume :
- 44
- Database :
- OpenAIRE
- Journal :
- Journal of Medicinal Chemistry
- Accession number :
- edsair.doi.dedup.....b279d8dfae9cc7e30e290d2c1c70d132
- Full Text :
- https://doi.org/10.1021/jm0108505