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Soluble Polymer-Supported Synthesis of 5-Arylidene Thiazolidinones and Pyrimidinones Using a Novel Traceless Linker Strategy

Authors :
Xin Wang
Zhang Liu
Yue Huang
Lanping Ma
Jingkang Shen
Wei Zhang
Jia Li
Jing-Ya Li
Source :
Journal of Combinatorial Chemistry. 10:632-636
Publication Year :
2008
Publisher :
American Chemical Society (ACS), 2008.

Abstract

An efficient method for the soluble polymer-supported synthesis of 5-arylidene thiazolidinones and pyrimidinones using aniline as a traceless linker was described. Aldehyde substrates were attached to the polyethylene glycol (PEG)-bound aniline via an imine linkage, and after the subsequent PEG-promoted Suzuki coupling reaction for the diversification, Knoevenagel condensation was readily employed as the cleavage strategy.

Details

ISSN :
15204774 and 15204766
Volume :
10
Database :
OpenAIRE
Journal :
Journal of Combinatorial Chemistry
Accession number :
edsair.doi.dedup.....91a5e376771d1767bc15c71ae352e5b3