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Synthesis of base-substituted uridine 5'-phosphonate analogues as potential P2Y2 receptor ligands

Authors :
T. Kendall Harden
Serge Van Calenbergh
Matthew O. Barrett
Kenneth A. Jacobson
Sara Van Poecke
Hocek, Michal
Source :
Collection Symposium
Publication Year :
2011
Publisher :
Academy of Sciences of the Czech Republic. Institute of Organic Chemistry and Biochemsitry, 2011.

Abstract

A series of 5-modified 5’-phosphonate derivatives of UMP has been prepared in 6 steps from uridine. The analogs were evaluated for their affinity at the P2Y2 receptor. Several derivatives showed partial agonistic activity at the P2Y2 receptor.

Details

Language :
English
ISBN :
978-80-86241-37-1
ISBNs :
9788086241371
Database :
OpenAIRE
Journal :
Collection Symposium
Accession number :
edsair.doi.dedup.....54c937f27ec3b6ee4dff0e4478bcf8e3