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Characterization of JNJ-2482272 [4-(4-Methyl-2-(4-(Trifluoromethyl)Phenyl)Thiazole-5-yl) Pyrimidine-2-Amine] As a Strong Aryl Hydrocarbon Receptor Activator in Rat and Human
- Source :
- Drug metabolism and disposition: the biological fate of chemicals. 50(8)
- Publication Year :
- 2021
-
Abstract
- [4-(4-Methyl-2-(4-(trifluoromethyl)phenyl)thiazole-5-yl)pyrimidine-2-amine] (JNJ-2482272), under investigation as an anti-inflammatory agent, was orally administered to rats once daily at 60 mg/kg for 6 consecutive days. Despite high plasma exposure after single administration (C
Details
- ISSN :
- 1521009X
- Volume :
- 50
- Issue :
- 8
- Database :
- OpenAIRE
- Journal :
- Drug metabolism and disposition: the biological fate of chemicals
- Accession number :
- edsair.doi.dedup.....4e7ffacc86d3af23c0c9e8fefda12a2a