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d4TMP Delivery from 7-SubstitutedcycloSal-d4TMPs

Authors :
Jan Balzarini
J. T. Renze
Chris Meier
E. De Clercq
Source :
Nucleosides, Nucleotides and Nucleic Acids. 22:825-827
Publication Year :
2003
Publisher :
Informa UK Limited, 2003.

Abstract

Benzyl-substituted cycloSal-d4T monophosphates were prepared and evaluated for their ability to release d4TMP selectively. In contrast to previously reported derivatives, two of the new compounds release d4TMP as the sole product while two others gave the expected benzyl phosphate diesters. However, these diesters were surprisingly stable against degradation to release d4TMP.

Details

ISSN :
15322335 and 15257770
Volume :
22
Database :
OpenAIRE
Journal :
Nucleosides, Nucleotides and Nucleic Acids
Accession number :
edsair.doi.dedup.....49d3ca1cb9c64962ffa11b9064d575d1
Full Text :
https://doi.org/10.1081/ncn-120022663