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Supplementary Methods from Preclinical Efficacy of the Novel Monocarboxylate Transporter 1 Inhibitor BAY-8002 and Associated Markers of Resistance

Authors :
Andrea Hägebarth
Marcus Bauser
Holger Siebeneicher
Atanas Kamburov
Ralf Lesche
Claudia Merz
Joern Toedling
Carmen Richter
Roland Neuhaus
Luisella Toschi
Ashley Eheim
Wolfgang Schwede
Andreas Schlicker
Sylvia Grünewald
Charlotte Kopitz
Eckhard Bender
Maria Quanz
Publication Year :
2023
Publisher :
American Association for Cancer Research (AACR), 2023.

Abstract

Supplementary Methods: Synthesis and characterization of BAY-8002; Tritium labeling of AZD3965 and BAY-8002; MCT1 and MCT4 14C-lactate uptake measurements in the X. laevis oocytes expression System

Details

Database :
OpenAIRE
Accession number :
edsair.doi.dedup.....2b9c449390e8d6d58b8fd14c10da3442
Full Text :
https://doi.org/10.1158/1535-7163.22505181