UR-DEBa242: A Py-5-Labeled Fluorescent Multipurpose Probe for Investigations on the Histamine H3 and H4 Receptors

Authors :: Ulla Seibel
Günther Bernhardt
David Wifling
Timo Littmann
Edith Bartole
Lukas Grätz
Armin Buschauer
Source :: Journal of Medicinal Chemistry. 63:5297-5311
Publication Year :: 2020
Publisher :: American Chemical Society (ACS), 2020.
Abstract: Comprehensively characterized fluorescent probes for the histamine H3 receptor (H3R) and especially for the H4R orthologs [e.g., human (h) and mouse (m)] are highly needed as versatile complementar...

Subjects :: 0303 health sciences
Chemistry
01 natural sciences
Fluorescence
0104 chemical sciences
010404 medicinal & biomolecular chemistry
03 medical and health sciences
chemistry.chemical_compound
Biochemistry
Drug Discovery
Molecular Medicine
Histamine H3 receptor
Receptor
Histamine
030304 developmental biology

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