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Conversion of NSAIDS into balanced dual inhibitors of cyclooxygenase and 5-lipoxygenase

Authors :
Dirk A. Bornemeier
David T. Connor
Diane H. Boschelli
Milton L. Hoefle
Richard D. Dyer
Source :
Bioorganic & Medicinal Chemistry Letters. 2:69-72
Publication Year :
1992
Publisher :
Elsevier BV, 1992.

Abstract

By replacing the carboxylic acid functionality of several fenamates with 1,3,4-oxadiazole-2-thiones and 1,3,4-thiadiazole-2-thiones we converted selective cycloxygenase (CO) inhibitors ito dual inhibitors of both CO and 5-lipoxygenase (5-LO).

Details

ISSN :
0960894X
Volume :
2
Database :
OpenAIRE
Journal :
Bioorganic & Medicinal Chemistry Letters
Accession number :
edsair.doi...........b52c84813e12191fad55054145533988
Full Text :
https://doi.org/10.1016/s0960-894x(00)80657-5