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Synthesis and Biological Evaluation of Furano-Epothilone C

Authors :
Dieter Schinzer
Karl-Heinz Altmann
Markus Wartmann
Oliver M. Böhm
Source :
Synlett. :1375-1378
Publication Year :
2004
Publisher :
Georg Thieme Verlag KG, 2004.

Abstract

An efficient synthesis of furano-epothilone C (1) is described by the use of an aldol reaction and a ring-closing metathesis (RCM) for the closure of the macrocyclic ring system. This new type of analog contains a furan ring in the C8-C10 region of the macrocycle. The biology of this new class of epothilone C analog has been studied.

Details

ISSN :
14372096 and 09365214
Database :
OpenAIRE
Journal :
Synlett
Accession number :
edsair.doi...........11b13f0cc3a12812d0e85622a9d958b6
Full Text :
https://doi.org/10.1055/s-2004-829071