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Discovery of antibacterial agents targeting biofilm formation: total synthesis and in vitro investigation of amycolasporins

Authors :
Wenxi Wu
Yu Mu
Junfeng Tan
Zixuan Wang
Chen Zhang
Guiding Li
Ying Jin
Xueshi Huang
Li Han
Source :
Organic & Biomolecular Chemistry. 20:6831-6843
Publication Year :
2022
Publisher :
Royal Society of Chemistry (RSC), 2022.

Abstract

The total synthesis of antibacterial amycolasporin A, (±) amycolasporins B and C and their analogues (18, 19, 30a and 30d–30f) was introduced; 30d obviously inhibited bacterial biofilm formation and promoted intracellular ROS release.

Details

ISSN :
14770539 and 14770520
Volume :
20
Database :
OpenAIRE
Journal :
Organic & Biomolecular Chemistry
Accession number :
edsair.doi...........0c04c24655fbdc25a175feb014cb9430
Full Text :
https://doi.org/10.1039/d2ob01166b