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A Practical Method for the Synthesis of a Cyclosporine−Fluorescein Conjugate

Authors :
Grote, J.
Fishpaugh, J.
Rege, S.
Source :
Organic Process Research & Development; November 2005, Vol. 9 Issue: 6 p822-824, 3p
Publication Year :
2005

Abstract

A straightforward synthesis of a cyclosporine−fluorescein conjugate through the MeBmt hydroxyl group was developed. Reaction of cyclosporine A in phosgene/toluene solution with added triethylamine, followed by subsequent reaction with 4‘-aminomethylfluorescein, produces good yields of the cyclosporine−fluorescein conjugate.

Details

Language :
English
ISSN :
10836160 and 1520586X
Volume :
9
Issue :
6
Database :
Supplemental Index
Journal :
Organic Process Research & Development
Publication Type :
Periodical
Accession number :
ejs8150325