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Discoveryof 1-[3-(1-Methyl-1H-pyrazol-4-yl)-5-oxo-5H-benzo[4,5]cyclohepta[1,2-b]pyridin-7-yl]-N-(pyridin-2-ylmethyl)methanesulfonamide(MK-8033): A Specific c-Met/Ron Dual Kinase Inhibitor withPreferential Affinity for the Activated State of c-Met.

Details

Language :
English
ISSN :
00222623
Volume :
56
Issue :
6
Database :
Supplemental Index
Journal :
Journal of Medicinal Chemistry
Publication Type :
Academic Journal
Accession number :
86450028
Full Text :
https://doi.org/10.1021/jm301619u