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Discoveryof 1-[3-(1-Methyl-1H-pyrazol-4-yl)-5-oxo-5H-benzo[4,5]cyclohepta[1,2-b]pyridin-7-yl]-N-(pyridin-2-ylmethyl)methanesulfonamide(MK-8033): A Specific c-Met/Ron Dual Kinase Inhibitor withPreferential Affinity for the Activated State of c-Met.
- Source :
- Journal of Medicinal Chemistry; Vol. 56 Issue 6, p2294-2310, 17p
- Publication Year :
- 2013
Details
- Language :
- English
- ISSN :
- 00222623
- Volume :
- 56
- Issue :
- 6
- Database :
- Supplemental Index
- Journal :
- Journal of Medicinal Chemistry
- Publication Type :
- Academic Journal
- Accession number :
- 86450028
- Full Text :
- https://doi.org/10.1021/jm301619u