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Design, Synthesis, and Pharmacodynamic Evaluation of Highly Selective PARP1 Inhibitors with Brain Penetrance.

Authors :
Guo, Tao
Yuan, Yongting
Zou, Yurong
Guo, Zhongning
Yang, Tao
Tang, Minghai
Ma, Ziyan
Fu, Zhiyuan
Bo, Weichen
Wang, Peng
Bai, Peng
Wang, Taijin
Jia, Tao
Yang, Jianhong
Chen, Lijuan
Source :
Journal of Medicinal Chemistry; 1/23/2025, Vol. 68 Issue 2, p1731-1754, 24p
Publication Year :
2025

Details

Language :
English
ISSN :
00222623
Volume :
68
Issue :
2
Database :
Supplemental Index
Journal :
Journal of Medicinal Chemistry
Publication Type :
Academic Journal
Accession number :
182440609
Full Text :
https://doi.org/10.1021/acs.jmedchem.4c02463