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Optimization of P2Y12 Antagonist Ethyl 6‑(4-((Benzylsulfonyl)carbamoyl)piperidin-1-yl)-5-cyano-2-methylnicotinate (AZD1283) Led to the Discovery of an Oral Antiplatelet Agent with Improved Druglike Properties.
- Source :
- Journal of Medicinal Chemistry; 3/28/2019, Vol. 62 Issue 6, p3088-3106, 19p
- Publication Year :
- 2019
Details
- Language :
- English
- ISSN :
- 00222623
- Volume :
- 62
- Issue :
- 6
- Database :
- Supplemental Index
- Journal :
- Journal of Medicinal Chemistry
- Publication Type :
- Academic Journal
- Accession number :
- 151167346
- Full Text :
- https://doi.org/10.1021/acs.jmedchem.8b01971