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Discovery and Structure-Guided Optimization of Diarylmethanesulfonamide Disrupters of Glucokinase-Glucokinase Regulatory Protein (GK-GKRP) Binding: Strategic Use of a N → S (nN → s*S-X) Interaction for Conformational...

Details

Language :
English
ISSN :
00222623
Volume :
58
Issue :
24
Database :
Supplemental Index
Journal :
Journal of Medicinal Chemistry
Publication Type :
Academic Journal
Accession number :
113302686
Full Text :
https://doi.org/10.1021/acs.jmedchem.5b01367