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4-((R)-2-{[6-((S)-3-Methoxypyrrolidin-1-yl)-2-phenylpyrimidine-4-carbonyl]amino}-3-phosphonopropionyl)piperazine-1-carboxylic Acid Butyl Ester (ACT-246475) and Its Prodrug (ACT-281959), a Novel P2Y12 Receptor Antagonist with a Wider...

Authors :
Caroff, Eva
Hubler, Francis
Meyer, Emmanuel
Renneberg, Dorte
Gnerre, Carmela
Treiber, Alexander
Rey, Markus
Hess, Patrick
Steiner, Beat
Hilpert, Kurt
Riederer, Markus A.
Source :
Journal of Medicinal Chemistry; Dec2015, Vol. 58 Issue 23, p9133-9153, 21p
Publication Year :
2015

Details

Language :
English
ISSN :
00222623
Volume :
58
Issue :
23
Database :
Supplemental Index
Journal :
Journal of Medicinal Chemistry
Publication Type :
Academic Journal
Accession number :
113302649
Full Text :
https://doi.org/10.1021/acs.jmedchem.5b00933