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SAR Studies on TetrahydroisoquinolineDerivatives:The Role of Flexibility and Bioisosterism To Raise Potency and Selectivitytoward P-glycoprotein.

Authors :
Capparelli, Elena
Zinzi, Laura
Cantore, Mariangela
Contino, Marialessandra
Perrone, Maria Grazia
Luurtsema, Gert
Berardi, Francesco
Perrone, Roberto
Colabufo, Nicola A.
Source :
Journal of Medicinal Chemistry; Dec2014, Vol. 57 Issue 23, p9983-9994, 12p
Publication Year :
2014

Details

Language :
English
ISSN :
00222623
Volume :
57
Issue :
23
Database :
Supplemental Index
Journal :
Journal of Medicinal Chemistry
Publication Type :
Academic Journal
Accession number :
100137630
Full Text :
https://doi.org/10.1021/jm501640e