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New generation dopaminergic agents. 2. Discovery of 3-OH-phenoxyethylamine and 3-OH-N1-phenylpiperazine dopaminergic templates.

Authors :
Mewshaw RE
Husbands M
Gildersleeve ES
Webb MB
Shi X
Mazandarani H
Cockett MI
Ochalski R
Brennan JA
Abou-Gharbia M
Marquis K
McGaughey GB
Coupet J
Andree TH
Source :
Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 1998 Feb 03; Vol. 8 (3), pp. 295-300.
Publication Year :
1998

Abstract

Described in this report is a systematic study which led to the identification of two new dopamine D2 partial agonists (5 and 17). Phenols 5 and 17 represent prototypes of two new classes of D2 partial agonists as well as templates for the future design of novel dopaminergic agents.

Details

Language :
English
ISSN :
0960-894X
Volume :
8
Issue :
3
Database :
MEDLINE
Journal :
Bioorganic & medicinal chemistry letters
Publication Type :
Academic Journal
Accession number :
9871673
Full Text :
https://doi.org/10.1016/s0960-894x(98)00014-6