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Palladium-Catalyzed Regioselective Synthesis of 2-SF 5 -Indenols and Further Derivatizations.

Authors :
Popek L
Cihan M
Blanchard N
Bizet V
Source :
Angewandte Chemie (International ed. in English) [Angew Chem Int Ed Engl] 2024 Feb 12; Vol. 63 (7), pp. e202315909. Date of Electronic Publication: 2024 Jan 11.
Publication Year :
2024

Abstract

A palladium-catalyzed synthesis of 2-SF <subscript>5</subscript> -indenols has been developed by reacting commercially available boronic acid derivatives and readily accessible SF <subscript>5</subscript> -alkynes. The present methodology is fully regioselective thanks to the intrinsic polarization of SF <subscript>5</subscript> -alkynes. A selection of downstream functionalizations has been performed to highlight the versatility of 2-SF <subscript>5</subscript> -indenols and indenones as platforms for the design of more complex SF <subscript>5</subscript> -containing molecules.<br /> (© 2023 The Authors. Angewandte Chemie International Edition published by Wiley-VCH GmbH.)

Details

Language :
English
ISSN :
1521-3773
Volume :
63
Issue :
7
Database :
MEDLINE
Journal :
Angewandte Chemie (International ed. in English)
Publication Type :
Academic Journal
Accession number :
38116823
Full Text :
https://doi.org/10.1002/anie.202315909