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Piperic acid derivative as a molecular modulator to accelerate the IAPP aggregation process and alter its antimicrobial activity.

Authors :
Chan AC
Shan PY
Wu MH
Lin PH
Tsai CS
Hsu CC
Chiu TH
Hsu TW
Yeh YC
Lai YJ
Liu WM
Tu LH
Source :
Chemical communications (Cambridge, England) [Chem Commun (Camb)] 2023 Aug 31; Vol. 59 (71), pp. 10660-10663. Date of Electronic Publication: 2023 Aug 31.
Publication Year :
2023

Abstract

Piperic acid derivatives were found to affect the islet amyloid polypeptide (IAPP) aggregation process. Structure-activity relationship studies revealed that PAD-13 was an efficient molecular modulator to accelerate IAPP fibril formation by promoting primary and secondary nucleation and reducing its antimicrobial activity.

Details

Language :
English
ISSN :
1364-548X
Volume :
59
Issue :
71
Database :
MEDLINE
Journal :
Chemical communications (Cambridge, England)
Publication Type :
Academic Journal
Accession number :
37581279
Full Text :
https://doi.org/10.1039/d3cc03363e