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Copper-Catalyzed Vicinal Cyano-, Thiocyano-, and Chlorophosphorylation of Alkynes: A Phosphinoyl Radical-Initiated Approach for Difunctionalized Alkenes.

Authors :
Tao ZK
Li CK
Li JA
Shoberu A
Zhang W
Zou JP
Source :
Organic letters [Org Lett] 2021 Jun 04; Vol. 23 (11), pp. 4342-4347. Date of Electronic Publication: 2021 May 24.
Publication Year :
2021

Abstract

A copper-catalyzed difunctional cyano-, thiocyano-, and chlorophosphorylation reaction of alkynes with P(O)-H compounds and coupling partners (TBACN, TMSNCS, TMSCl) is described. The reaction introduces versatile groups (-P(O)R <subscript>2</subscript> and -CN, -SCN, or -Cl) to form tri- and tetrasubstituted alkenyl phosphine oxides/phosphonates regio- and stereoselectively.

Details

Language :
English
ISSN :
1523-7052
Volume :
23
Issue :
11
Database :
MEDLINE
Journal :
Organic letters
Publication Type :
Academic Journal
Accession number :
34029107
Full Text :
https://doi.org/10.1021/acs.orglett.1c01286