Back to Search Start Over

Palladium-Catalyzed Amination/Dearomatization Reaction of Indoles and Benzofurans.

Authors :
Zhang Z
Zhang BS
Li KL
An Y
Liu C
Gou XY
Liang YM
Source :
The Journal of organic chemistry [J Org Chem] 2020 Jun 19; Vol. 85 (12), pp. 7817-7839. Date of Electronic Publication: 2020 Jun 01.
Publication Year :
2020

Abstract

This report describes a palladium-catalyzed dearomatization and amination tandem reaction of 2,3-disubstituted indoles and benzofurans via the Catellani strategy. This reaction provides a new method for the construction of amino-substituted indoline-fused cyclic and benzofuran spiro compounds in good yields. The reaction has broad functional group compatibility and substrate scope.

Details

Language :
English
ISSN :
1520-6904
Volume :
85
Issue :
12
Database :
MEDLINE
Journal :
The Journal of organic chemistry
Publication Type :
Academic Journal
Accession number :
32441518
Full Text :
https://doi.org/10.1021/acs.joc.0c00475