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Methodology for Identification of Cysteine-Reactive Covalent Inhibitors.

Authors :
Kathman SG
Statsyuk AV
Source :
Methods in molecular biology (Clifton, N.J.) [Methods Mol Biol] 2019; Vol. 1967, pp. 245-262.
Publication Year :
2019

Abstract

Covalent fragments are an emerging technology to discover covalent ligands in target-based or phenotypic screens. Here we describe screening of cysteine-reactive covalent fragments against a protein of interest using mass spectrometry or enzymatic methods.

Details

Language :
English
ISSN :
1940-6029
Volume :
1967
Database :
MEDLINE
Journal :
Methods in molecular biology (Clifton, N.J.)
Publication Type :
Academic Journal
Accession number :
31069775
Full Text :
https://doi.org/10.1007/978-1-4939-9187-7_15