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Copper-Catalyzed Oxidative sp 3 -Carbon Radical Cross-Coupling with Trialkylphosphites Leading to α-Phosphonyl 1,3-Dicarbonyl Compounds.

Authors :
Li CK
Tao ZK
Zhou ZH
Bao XG
Zhou SF
Zou JP
Source :
The Journal of organic chemistry [J Org Chem] 2019 Feb 15; Vol. 84 (4), pp. 2351-2357. Date of Electronic Publication: 2019 Feb 04.
Publication Year :
2019

Abstract

A copper-catalyzed radical C <subscript>sp <superscript>3</superscript> </subscript> -H/P(OR) <subscript>3</subscript> cross-coupling reaction for the formation of C <subscript>sp <superscript>3</superscript> </subscript> -P bonds is described. A range of 1,3-dicarbonyl compounds and trialkylphosphites were coupled in this fashion to give the corresponding products in moderate to good yields. This protocol provides direct access to α-phosphonyl 1,3-dicarbonyl compounds.

Details

Language :
English
ISSN :
1520-6904
Volume :
84
Issue :
4
Database :
MEDLINE
Journal :
The Journal of organic chemistry
Publication Type :
Academic Journal
Accession number :
30667228
Full Text :
https://doi.org/10.1021/acs.joc.8b03093