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Metal-Free Formal Inverse-Electron-Demand Diels-Alder Reaction of 1,2-Diazines with Ynamides.

Authors :
Xue J
Gao E
Wang XN
Chang J
Source :
Organic letters [Org Lett] 2018 Oct 05; Vol. 20 (19), pp. 6055-6058. Date of Electronic Publication: 2018 Sep 20.
Publication Year :
2018

Abstract

A highly effective metal-free formal inverse-electron-demand Diels-Alder reaction of 1,2-diazines with ynamides has been developed. This catalytic protocol is more environmentally friendly and allows for the construction of 2-aminonaphthalenes and 2-aminoanthracenes from 1,2-diazines and ynamides in good to high yields with wide diversity and functional group tolerance.

Details

Language :
English
ISSN :
1523-7052
Volume :
20
Issue :
19
Database :
MEDLINE
Journal :
Organic letters
Publication Type :
Academic Journal
Accession number :
30234310
Full Text :
https://doi.org/10.1021/acs.orglett.8b02431