Back to Search Start Over

Non-Directed Cross-Dehydrogenative (Hetero)arylation of Allylic C(sp 3 )-H bonds enabled by C-H Activation.

Authors :
Lerchen A
Knecht T
Koy M
Ernst JB
Bergander K
Daniliuc CG
Glorius F
Source :
Angewandte Chemie (International ed. in English) [Angew Chem Int Ed Engl] 2018 Nov 12; Vol. 57 (46), pp. 15248-15252. Date of Electronic Publication: 2018 Oct 12.
Publication Year :
2018

Abstract

Herein, we report the selective, non-directed and cross-dehydrogenative coupling of allylic C(sp <superscript>3</superscript> )-H bonds with C(sp <superscript>2</superscript> )-H bonds of (hetero)arenes. The methodology employs olefins and (hetero)arenes which are abundantly available chemical feedstocks, and could be applied in late-stage functionalization reactions of pharmaceuticals. Furthermore, the system exclusively delivers the allylic C-C coupling products highlighting the preservation of the olefin substitution pattern for further derivatization.<br /> (© 2018 Wiley-VCH Verlag GmbH & Co. KGaA, Weinheim.)

Details

Language :
English
ISSN :
1521-3773
Volume :
57
Issue :
46
Database :
MEDLINE
Journal :
Angewandte Chemie (International ed. in English)
Publication Type :
Academic Journal
Accession number :
30152920
Full Text :
https://doi.org/10.1002/anie.201807047