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Lipase catalyzed synthesis of antimicrobial andrographolide derivatives.

Authors :
Patil HS
Jadhav DD
Paul A
Mulani FA
Karegaonkar SJ
Thulasiram HV
Source :
Data in brief [Data Brief] 2018 Mar 28; Vol. 18, pp. 1134-1141. Date of Electronic Publication: 2018 Mar 28 (Print Publication: 2018).
Publication Year :
2018

Abstract

In this data article we describe screening of various lipases for the regioselective acylation of Andrographolide. Each lipase was screened with seven acyl donors. Amano lipase AK from Pseudomonas fluorescens was used for the synthesis of two new acylated andrographolide derivatives. Two new compounds, andrographolide-14-propionate and andrographolide-14-caproate were characterized by various spectral studies. These two derivatives showed more antimicrobial activity than andrographolide.

Details

Language :
English
ISSN :
2352-3409
Volume :
18
Database :
MEDLINE
Journal :
Data in brief
Publication Type :
Academic Journal
Accession number :
29900286
Full Text :
https://doi.org/10.1016/j.dib.2018.03.103