Back to Search Start Over

Palladium-Catalyzed One-Pot Approach to 3-(Diarylmethylene)oxindoles from Propiolamidoaryl Triflate.

Authors :
Lee D
Park S
Yu Y
Shin KJ
Seo JH
Source :
Molecules (Basel, Switzerland) [Molecules] 2015 Aug 03; Vol. 20 (8), pp. 14022-32. Date of Electronic Publication: 2015 Aug 03.
Publication Year :
2015

Abstract

3-(Diarylmethylene)oxindoles have been synthesized from propiolamidoaryl triflate utilizing a palladium-catalyzed one-pot reaction consisting of three successive reactions: Sonogashira, Heck, and Suzuki-Miyaura. This method allows for the production of a complex skeleton of 3-(diarylmethylene)oxindole from propiolamidoaryl triflate using a commercially available aryl iodide and arylboronic acid in a simple and efficient way with moderate yield and stereoselectivity.

Details

Language :
English
ISSN :
1420-3049
Volume :
20
Issue :
8
Database :
MEDLINE
Journal :
Molecules (Basel, Switzerland)
Publication Type :
Academic Journal
Accession number :
26247925
Full Text :
https://doi.org/10.3390/molecules200814022