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Zopolrestat as a human glyoxalase I inhibitor and its structural basis.
- Source :
-
ChemMedChem [ChemMedChem] 2013 Sep; Vol. 8 (9), pp. 1462-4. Date of Electronic Publication: 2013 Jul 15. - Publication Year :
- 2013
- Subjects :
- Animals
Anti-Inflammatory Agents, Non-Steroidal metabolism
Benzothiazoles metabolism
Binding Sites
Crystallography, X-Ray
Enzyme Inhibitors metabolism
Humans
Indomethacin chemistry
Indomethacin metabolism
Lactoylglutathione Lyase metabolism
Mice
Phthalazines metabolism
Protein Binding
Protein Structure, Tertiary
Anti-Inflammatory Agents, Non-Steroidal chemistry
Benzothiazoles chemistry
Enzyme Inhibitors chemistry
Lactoylglutathione Lyase chemistry
Phthalazines chemistry
Subjects
Details
- Language :
- English
- ISSN :
- 1860-7187
- Volume :
- 8
- Issue :
- 9
- Database :
- MEDLINE
- Journal :
- ChemMedChem
- Publication Type :
- Academic Journal
- Accession number :
- 23857942
- Full Text :
- https://doi.org/10.1002/cmdc.201300243