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Stereoselective hydrofluorination of ynamides: a straightforward synthesis of novel α-fluoroenamides.

Authors :
Compain G
Jouvin K
Martin-Mingot A
Evano G
Marrot J
Thibaudeau S
Source :
Chemical communications (Cambridge, England) [Chem Commun (Camb)] 2012 May 25; Vol. 48 (42), pp. 5196-8. Date of Electronic Publication: 2012 Apr 18.
Publication Year :
2012

Abstract

α-Fluoroenamides, potent rigid fluorinated bioisosters of ureas, have been synthesized by a highly regio- and stereo-selective hydrofluorination of ynamides in anhydrous HF. This reaction provides the first general entry to α-fluoroenamides and can easily be applied to a wide range of substrates.<br /> (This journal is © The Royal Society of Chemistry 2012)

Details

Language :
English
ISSN :
1364-548X
Volume :
48
Issue :
42
Database :
MEDLINE
Journal :
Chemical communications (Cambridge, England)
Publication Type :
Academic Journal
Accession number :
22514037
Full Text :
https://doi.org/10.1039/c2cc31768k