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Synthesis of purine modified 2'-C-methyl nucleosides as potential anti-HCV agents.

Authors :
Zhang HW
Zhou L
Coats SJ
McBrayer TR
Tharnish PM
Bondada L
Detorio M
Amichai SA
Johns MD
Whitaker T
Schinazi RF
Source :
Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2011 Nov 15; Vol. 21 (22), pp. 6788-92. Date of Electronic Publication: 2011 Sep 20.
Publication Year :
2011

Abstract

Based on the anti-hepatitis C activity of 2'-C-methyl-adenosine and 2'-C-methyl-guanosine, a series of new modified purine 2'-C-methyl nucleosides was prepared as potential anti-hepatitis C virus agents. Herein, we report the synthesis of both 6-modified and 2-modified purine 2'-C-methyl-nucleosides along with their anti-HCV replication activity and cytotoxicity in different cells.<br /> (Published by Elsevier Ltd.)

Details

Language :
English
ISSN :
1464-3405
Volume :
21
Issue :
22
Database :
MEDLINE
Journal :
Bioorganic & medicinal chemistry letters
Publication Type :
Academic Journal
Accession number :
21983447
Full Text :
https://doi.org/10.1016/j.bmcl.2011.09.034