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Pentamidine Congeners 1: Synthesis of Cis- and Trans-Butamidine Analogues As Anti-Pneumocystis carinii Pneumonia Agents.

Authors :
Donkor IO
Jones SK
Tidwell RR
Source :
Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 1993; Vol. 3 (6), pp. 1137-1140.
Publication Year :
1993

Abstract

Butamidine analogues possessing unsaturation in the ether bridge between the bisamidinophenyl or bisimidazolinophenyl functionalities have been synthesized as semirigid congeners of pentamidine. These compounds demonstrated good anti-P. carinii pueumonia activity in a rat model of the disease.

Details

Language :
English
ISSN :
1464-3405
Volume :
3
Issue :
6
Database :
MEDLINE
Journal :
Bioorganic & medicinal chemistry letters
Publication Type :
Academic Journal
Accession number :
21451734
Full Text :
https://doi.org/10.1016/S0960-894X(00)80302-9