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Synthesis of novel cholesterol-based cationic lipids for gene delivery.

Authors :
Kim BK
Doh KO
Nam JH
Kang H
Park JG
Moon IJ
Seu YB
Source :
Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2009 Jun 01; Vol. 19 (11), pp. 2986-9. Date of Electronic Publication: 2009 Apr 18.
Publication Year :
2009

Abstract

The new cholesterol-based cationic lipids B, C, and D with an ether linked spacer were synthesized by using aminopropyl chain extension with acrylonitrile. The cholesterol-based cationic lipid A with carbamoyl linkage were also synthesized in order to compare the difference in transfection efficiency of the two linkage types. To this end, GFP expression of these cationic lipids was confirmed respectively.

Details

Language :
English
ISSN :
1464-3405
Volume :
19
Issue :
11
Database :
MEDLINE
Journal :
Bioorganic & medicinal chemistry letters
Publication Type :
Academic Journal
Accession number :
19409781
Full Text :
https://doi.org/10.1016/j.bmcl.2009.04.036